Novel Oral Analgesic Drug Tapentadol Hydrochloride CAS 175591-09-0

Basic Info

Model No.: 175591-09-0

Additional Info

Packaging: As Quantity

Productivity: As Order

Brand: VOLSENCHEM

Transportation: Air

Place of Origin: CHINA

Supply Ability: IN STOCK

Product Description

Tapentadol Hydrochloride CAS Number is 175591-09-0, tapentadol hydrochloride is a novel oral analgesic drug acting on the central nervous system. It has two mechanisms of action: one is acting on the opioid μ2 receptor. By improving pain sensation and affective factors, inhibiting the transmission of pain in the spinal cord, thereby affecting and controlling the activity of the cerebral cortex that senses pain; the other is the inhibition of norepinephrine reuptake, inhibiting its reabsorption into the nerve The cells, which raise the level of norepinephrine in the brain, also serve as an analgesic effect. Tapentadol hydrochloride does not rely on metabolic activation, no metabolic activation products, and has a strong effect on various acute inflammations and neuralgia. Both intravenous and oral administration can achieve higher blood concentration, and it is not easy to produce analgesic resistance and dependence.
Tapentadol Hydrochloride CAS Number 175591-09-0 is a central analgesic developed by Gruenenthal and Johnson & Johnson in Germany. It has the dual role of opioid μ receptor agonist and adrenergic transmitter uptake inhibitor. It was acquired on November 21, 2008 in the United States. The FDA is approved for marketing and is used clinically to relieve moderate to severe acute pain in adults.Tapentadol Hydrochloride CAS 175591-09-0 is more tolerant and less toxic than other opioid analgesics.

Thera. Category:Anti- analgesic 

Cas No.: 175591-09-0

Synonyms:3-[(1R,2R)-3-(Dimethylamino)-1-ethyl-2-methylpropyl]phenol Hydrochloride;Tapentadol Hydrochloride;Tapentadol hcl;Phenol, 3-[(1R,2R)-3-(diMethylaMino)-1-ethyl-2-Methylpropyl]-,( 57202382,HCl salt);3-[(1R,2R)-3-(DiMethylaMino)-1-ethyl-2-Methylpro;3-((2R,3R)-1-(diMethylaMino)-2-Methylpentan-3-yl)phenol hydrochloride;Phenol,3-[(1R,2R)-3-(diMethylaMino)-1-ethyl-2-Methylpropyl]-, hydrochloride (1:1);Tapentadol hydrochloride solution

MF:  C14H24ClNO

NW:257.81

Assay: ≥99%

Packing:Export worthy packing

Material Safety Data Sheet:Available on request